Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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1,306
Tocris Bioscience™ CGP 71683 hydrochloride
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Highly selective and potent non-peptide NPY Y5 receptor antagonist
| Inhibitors | CGP 71683 hydrochloride |
|---|---|
| Product Type | CGP 71683 hydrochloride |
| Molecular Weight (g/mol) | 512.07 |
| Purity | >99% |
1,307
Tocris Bioscience™ IT1t dihydrochloride
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CAS: 1092776-63-0 Molecular Formula: C21H36Cl2N4S2
| CAS | 1092776-63-0 |
|---|---|
| Molecular Formula | C21H36Cl2N4S2 |
1,308
Tocris Bioscience™ SCIO 469 hydrochloride
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CAS: 309913-83-5 Molecular Formula: C27H30ClFN4O3
| CAS | 309913-83-5 |
|---|---|
| Molecular Formula | C27H30ClFN4O3 |
1,309
Tocris Bioscience™ IB-MECA
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CAS: 152918-18-8 Molecular Formula: C18H19IN6O4
| CAS | 152918-18-8 |
|---|---|
| Molecular Formula | C18H19IN6O4 |
1,310
Tocris Bioscience™ 27-Hydroxycholesterol
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LXR agonist; also ER partial agonist
1,311
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Tocris Bioscience™ C25-140
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Tocris Bioscience™ C25-140
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TRAF6-Ubc13 interaction inhibitor
| Target | Ubiquitin Ligase (E3) Inhibitors |
|---|---|
| CAS | 1358099-18-9 |
| Chemical Name or Material | 3-[3,5-Dimethyl-1-(3-methyl-1,2,4-triazolo[4,3-b]pyridazin-6-yl)-1H-pyrazol-4-yl]-1-[4-(phenylmethyl)-1-piperidinyl]-1-propanone |
| Recommended Storage | Store the unopened product at -20 to -70 °C. Use a manual defrost freezer and avoid repeated freeze-thaw cycles. Do not use past expiration date. |
| Molecular Formula | C26H31N7O |
1,312
Tocris Bioscience™ BIBN 4096
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Small and Specialty Supplier Partner
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Potent and selective CGRP antagonist
1,313
Tocris Bioscience™ OXA 06 dihydrochloride
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent ROCK inhibitor
| Inhibitors | OXA 06 dihydrochloride |
|---|---|
| CAS | 1825455-91-1 |
| Product Type | OXA 06 dihydrochloride |
| Molecular Weight (g/mol) | 404.31 |
| Purity | >98% |
1,314
Tocris Bioscience™ Ceritinib
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Highly potent ALK inhibitor; also potently inhibits IR, IGF1R, STK22D and FLT3
| Product Type | Inhibitor |
|---|---|
| Purity | 98% |
| Recommended Storage | Store at 4°C |
| Synonym | LDK378 |
| Molecular Formula | C28H36ClN5O3S |
| Formula Weight | 558.14 |
1,315
Tocris Bioscience™ Lalistat 2
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Selective LAL inhibitor
| CAS | 1234569-09-5 |
|---|---|
| Chemical Name or Material | 4-(Piperidin-1-yl)-1,2,5-thiadiazol-3-yl piperidine-1-carboxylate |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C13H20N4O2S |
| Formula Weight | Observed MW: 296.39 |
| Assay Percent Range | >98% |
1,316
Tocris Bioscience™ SAG
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Potent Smoothened receptor agonist; activates the Hedgehog signaling pathway
| Inhibitors | SAG |
|---|---|
| Product Type | SAG |
| Molecular Weight (g/mol) | 490.06 |
| Purity | >99% |
1,317
Tocris Bioscience™ KT 5823
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 126643-37-6 Molecular Formula: C29H25N3O5
| CAS | 126643-37-6 |
|---|---|
| Molecular Formula | C29H25N3O5 |
1,318
Tocris Bioscience™ trans-Ned 19
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CAS: 1354235-96-3 Molecular Formula: C30H31FN4O3
| CAS | 1354235-96-3 |
|---|---|
| Molecular Formula | C30H31FN4O3 |
1,319
Tocris Bioscience™ SB 334867
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Selective non-peptide OX1 antagonist
| CAS | 792173-99-0 |
|---|---|
| Solubility | Soluble to 100mM with gentle warming in DMSO |
| Chemical Name or Material | N-(2-Methyl-6-benzoxazolyl)-N'-1,5-naphthyridin-4-yl urea |
| Recommended Storage | Desiccate at Room Temperature |
| Molecular Formula | C17H13N5O2 |
| Formula Weight | Observed MW: 319.32 |
| Assay Percent Range | >99% |
1,320
Tocris Bioscience™ TC-S 7004
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Potent and selective DYRK1A/B inhibitor
| Product Type | TC-S 7004 |
|---|---|
| Molecular Weight (g/mol) | 498.32 |
| Purity | >98% |